Does Ketoconazole, Micronized (Bulk) 100 % Powder Interact with other Medications?
Severe Interactions
These medications are not usually taken together. Consult your healthcare professional (e.g., doctor or pharmacist) for more in formation.
- MISC ANTIFUNGAL AGENTS/ASTEMIZOLE; TERFENADINE
- ITRACONAZOL;KETOCONAZOL;LEVOKETOCONAZ/SLT BENZODIAZEPINES
- ITRACONAZOLE; KETOCONAZOLE; LEVOKETOCONAZOLE/ISONIAZID
- STRONG CYP3A4 INHIBITORS/GEPIRONE
- SELECTED STRONG AND MODERATE CYP3A4 INHIBITORS/CISAPRIDE
- STR 3A4 INHIB;ATAZAN;DARUN/COLCHICINE (FOR CARDIOPROTECTION)
- STR CYP3A4 INHIBITORS; PROTEASE INHIB/PIMAVANSERIN (> 10 MG)
- STRONG CYP3A4 INHIBITORS/MAVACAMTEN
- STRONG CYP3A4 INHIBITORS/PACRITINIB
- STRONG CYP3A4 INHIBITORS/DARIDOREXANT
- SELECTED STRONG CYP3A4 INHIBITORS/CONIVAPTAN
- SELECTED STRONG CYP3A4 INHIBITORS/ALFUZOSIN
- STRONG CYP3A4 INHIBITORS/FINERENONE
- STRONG CYP3A4 INHIBITORS/VOCLOSPORIN
- STRONG AND MODERATE CYP3A4 INHIBITORS/LONAFARNIB
- KETOCONAZOLE; POSACONAZOLE/SLT HMG-COA REDUCTASE INHIBITORS
- STRONG CYP3A4 INHIB; PROTEASE INHIB/LUMATEPERONE (>10.5 MG)
- STRONG CYP3A4 INHIBITORS/UBROGEPANT
- STRONG CYP3A4 INHIBITORS; ATAZANAVIR;DARUNAVIR/LERCANIDIPINE
- SLT STRONG & MODERATE CYP3A4 INHIBITORS/CILOSTAZOL (>50MG)
- STRONG CYP3A4 INHIBITORS/DAPAGLIFLOZIN-SAXAGLIPTIN-METFORMIN
- STRONG AND MODERATE CYP3A4 INHIBITORS/ASUNAPREVIR
- STRONG CYP3A4 INHIBITORS/VALBENAZINE (> 40 MG)
- STRONG OR MODERATE CYP3A4 INHIBITORS/LOMITAPIDE
- SELECTED STRONG CYP3A4 INHIBITORS/ISAVUCONAZONIUM
- STRONG CYP3A4 INHIBITORS/PANOBINOSTAT (> 10 MG)
- STRONG CYP3A4 INHIBITORS/NALOXEGOL
- STRONG CYP3A4 INHIBITORS; ATAZANAVIR; DARUNAVIR/AVANAFIL
- 3A4INHIB/DAPOXETINE;LEVOMILNACIPRAN(>80MG);VILAZODONE(>20MG)
- STRONG OR MODERATE CYP3A4 INHIBITORS/FLIBANSERIN
- STRONG CYP3A4 INHIBITORS/SLT HIGH STRENGTH ANTIMUSCARINICS
- SELECTED STRONG AND MODERATE CYP3A4 INHIBITORS/DOMPERIDONE
- STRONG CYP3A4 INHIBITORS; PROTEASE INHIBITORS/TICAGRELOR
- SELECTED AZOLE ANTIFUNGAL AGENTS/LURASIDONE
- KETOCONAZOLE; LEVOKETOCONAZOLE/MEFLOQUINE
- STRONG CYP3A4 INHIB;ATAZANAV;DARUNAVIR/SAXAGLIPTIN (>2.5 MG)
- STRONG CYP3A4 INHIBITORS; DARUNAVIR/DRONEDARONE
- ITRACONAZOL;KETOCONAZOL;LEVOKETOCON/FELODIPINE;NISOLDIPINE
- P-GP AND STRONG CYP3A4 INHIBITORS/RIVAROXABAN
- STRONG CYP3A4 INHIBITORS; PROTEASE INHIBITORS/RANOLAZINE
- STRONG CYP3A4 INHIBITORS/TOLVAPTAN
- STRONG CYP3A4 INHIBITORS; PROTEASE INHIBITORS/IVABRADINE
- STRONG CYP3A4 INHIBITORS/SILODOSIN; TAMSULOSIN
- ITRACONAZOLE;KETOCONAZO/LEVOMETHADONE;LEVOMETHADYL;METHADONE
- SELECTED CYP3A4 INHIBITORS/VARDENAFIL (> 5 MG)
- ITRACONAZOLE; KETOCONAZOLE/ERGOT ALKALOIDS
- STRONG CYP3A4 INHIBITORS; PROTEASE INHIBITORS/EPLERENONE
- STRONG CYP3A4 INHIBITORS/IRINOTECAN
- SELECTED AZOLE ANTIFUNGALS/ELETRIPTAN
- ITRACONAZOLE; KETOCONAZOLE(ORAL)/DOFETILIDE
- SELECTED AZOLE ANTIFUNGALS/DISOPYRAMIDE; QUINIDINE
- SELECTED AZOLE ANTIFUNGALS/PIMOZIDE
- ITRACONAZOLE; KETOCONAZOLE/SERTINDOLE
Serious Interactions
These medications may interact and cause very harmful effects. Consult your healthcare professional (e.g., doctor or pharmacist) for more in formation.
- ITRACONAZOLE; KETOCONAZOLE/DIGOXIN
- SELECT AZOLE ANTIFUNGAL AGENTS/COUMARIN ANTICOAGULANTS
- AZOLE ANTIFUNGAL AGENTS/SELECTED RIFAMYCINS
- ITRACONAZOLE; KETOCONAZOLE/NEVIRAPINE
- ITRACONAZOLE; KETOCONAZOLE; POSACONAZOLE/EFAVIRENZ
- AZOLE ANTIFUNGAL AGENTS/RIFABUTIN
- SELECTED AZOLE ANTIFUNGAL CYP3A4 SUBSTRATES/ENASIDENIB
- STRONG AND MODERATE CYP3A4 INHIBITORS/NIROGACESTAT
- STRONG CYP3A4 INHIBITORS/CAPIVASERTIB
- STRONG AND MODERATE CYP3A4 INHIBITORS/REPOTRECTINIB
- STRONG CYP3A4 OR MODERATE CYP2C9 INHIBITORS/ERDAFITINIB
- STRONG CYP3A4 INHIBITORS/REBOXETINE
- SELECTED CYP3A4 INHIBITORS/MEPERIDINE
- STRONG CYP3A4 INHIBITORS/PALOVAROTENE
- STRONG CYP3A4 INHIBITORS/TRETINOIN
- STRONG CYP3A4 INHIBITORS/LENIOLISIB
- STRONG CYP3A4 INHIBITORS/OMAVELOXOLONE
- STRONG CYP3A4 INHIBITORS/SPARSENTAN
- STRONG AND MODERATE CYP3A4 INHIBITORS/ELACESTRANT
- STRONG CYP3A4 INHIBITORS/PIRTOBRUTINIB
- STRONG CYP3A4 INHIBITORS/ADAGRASIB
- STRONG CYP3A4 INHIBITORS/PEXIDARTINIB
- DUAL STRONG CYP3A4 & P-GP INHIBITORS/FUTIBATINIB
- SELECTED STRONG CYP3A4 INHIBITORS/CLOZAPINE
- SELECTED AZOLE ANTIFUNGAL AGENTS/TACROLIMUS
- STRONG CYP3A4 INHIBITORS/MITAPIVAT
- STRONG CYP3A4 INHIBITOR/TOLTERODINE (>1 MG IR OR >2 MG ER)
- STRONG CYP3A4 INHIBITORS/RIVOCERANIB
- STRONG CYP3A4 INHIBITORS/LEVOKETOCONAZOLE
- STRONG CYP3A4 INHIBITORS/UPADACITINIB (>=30 MG)
- STRONG CYP3A4 INHIBITORS/RUPATADINE
- STRONG CYP3A4 INHIBITORS/SURUFATINIB
- STRONG CYP3A4 INHIBITORS/AVACOPAN
- STRONG CYP3A4 INHIBITORS/ATOGEPANT
- STRONG CYP3A4 INHIBITORS/MOBOCERTINIB
- UGT INHIBITORS/LORAZEPAM EXTENDED RELEASE
- STRONG AND MODERATE CYP3A4 INHIBITORS/FEXINIDAZOLE
- STRONG AND MODERATE CYP3A4 INHIBITORS/INFIGRATINIB
- P-GLYCOPROTEIN (P-GP) INHIBITORS/RELUGOLIX
- STRONG CYP3A4 INHIBITORS/TOREMIFENE
- STRONG CYP3A4 INHIBITORS/SUNITINIB
- STRONG CYP3A4 INHIBITORS/PAZOPANIB
- STRONG CYP3A4 INHIBITORS/NILOTINIB
- STRONG CYP3A4 INHIBITORS/LAPATINIB
- STRONG CYP3A4 INHIBITORS/DASATINIB
- STRONG CYP3A4 INHIBITORS/CRIZOTINIB
- STRONG CYP3A4 INHIBITORS/CERITINIB
- STRONG CYP3A4 INHIBITORS/VINFLUNINE
- STRONG CYP3A4 INHIBITORS/VINCRISTINE
- STRONG CYP3A4 INHIBITORS/VINBLASTINE
- STRONG CYP3A4 INHIBITORS/TOFACITINIB
- STRONG CYP3A4 INHIBITORS/SONIDEGIB
- STRONG CYP3A4 INHIBITORS/RUXOLITINIB
- STRONG CYP3A4 INHIBITORS/PONATINIB
- STRONG CYP3A4 INHIBITORS/PALBOCICLIB
- STRONG CYP3A4 INHIBITORS/PACLITAXEL
- STRONG CYP3A4 INHIBITORS/OLAPARIB
- STRONG CYP3A4 INHIBITORS/IXABEPILONE
- STRONG CYP3A4 INHIBITORS/IDELALISIB
- STRONG CYP3A4 INHIBITORS/ERLOTINIB
- STRONG CYP3A4 INHIBITORS/DOXORUBICIN
- STRONG CYP3A4 INHIBITORS/DOCETAXEL
- STRONG CYP3A4 INHIBITORS/DABRAFENIB
- STRONG CYP3A4 INHIBITORS/COBIMETINIB
- STRONG CYP3A4 INHIBITORS/CABOZANTINIB
- STRONG CYP3A4 INHIBITORS/CABAZITAXEL
- STRONG CYP3A4 INHIBITORS/AXITINIB
- STRONG CYP3A4 INHIBITORS; ATAZANAVIR; DARUNAVIR/SUVOREXANT
- DUAL STRONG CYP3A4 AND P-GP INHIBITORS/PRALSETINIB
- STRONG CYP3A4 INHIBITORS/PLITIDEPSIN
- KETOCONAZOLE; POSACONAZOLE/ATORVASTATIN
- STRONG CYP3A4 INHIBITORS/LURBINECTEDIN
- STRONG CYP3A4 INHIBITORS/SELPERCATINIB
- UGT1A1 INHIBITORS/SACITUZUMAB GOVITECAN
- STRONG AND MODERATE CYP3A4 INHIBITORS/PEMIGATINIB
- STRONG AND MODERATE CYP3A4 INHIBITORS/SELUMETINIB
- STRONG CYP3A4 INHIBITORS/RIMEGEPANT
- STRONG CYP3A4 INHIBITORS/NIMODIPINE
- STRONG CYP3A4 INHIBITORS/TAZEMETOSTAT
- STRONG CYP3A4 INHIBITORS/AVAPRITINIB
- SELECTED CYP3A4 INHIBITORS/SALMETEROL COMBINATIONS
- STRONG AND MODERATE CYP3A4 INHIBITORS/LEMBOREXANT
- STRONG CYP3A4 INHIBITORS/ELEXACAFTOR-TEZACAFTOR-IVACAFTOR
- STRONG CYP3A4 INHIBITORS/NALDEMEDINE
- STRONG CYP3A4 INHIBITORS/ISTRADEFYLLINE
- SELECTED STRONG CYP3A4 INHIBITORS/ORAL LEFAMULIN
- STRONG CYP3A4 INHIBITORS/FEDRATINIB
- STRONG CYP3A4 INHIBITORS/ENTRECTINIB
- STRONG CYP3A4 INHIBITORS/PEXIDARTINIB (200 MG)
- STRONG CYP3A4 INHIBITORS/BOSUTINIB
- SELECTED CYP3A4 INHIBITORS/ELBASVIR-GRAZOPREVIR
- STRONG CYP3A4 INHIBITORS/LAROTRECTINIB
- STRONG CYP3A4 INHIBITORS/GLASDEGIB
- STRONG CYP3A4 INHIBITORS/LORLATINIB
- STRONG CYP3A4 INHIBITORS/DUVELISIB
- STRONG CYP3A4 INHIBITORS/ELAGOLIX
- ITRACONAZOLE; KETOCONAZOLE/IVOSIDENIB
- STRONG CYP3A4 INHIBITORS/ARIPIPRAZOLE LAUROXIL SUBMICRONIZED
- STRONG AND MODERATE CYP3A4 INHIBITORS/ENCORAFENIB
- STRONG AND MODERATE CYP3A4 INHIBITORS/TEZACAFTOR-IVACAFTOR
- STRONG CYP3A4 INHIBITORS/IBRUTINIB
- STRONG CYP3A4 INHIBITORS/ACALABRUTINIB
- KETOCONAZOLE/ABEMACICLIB
- STRONG CYP3A4 INHIBITORS/COPANLISIB
- SELECTED P-GLYCOPROTEIN (P-GP) INHIBITORS/BETRIXABAN
- STRONG CYP3A4 INHIB;MODERATE 3A4 & P-GP DUAL INHIB/NERATINIB
- STRONG CYP3A4 INHIBITORS/BRIGATINIB
- STRONG CYP3A4 INHIBITORS/RIBOCICLIB
- STRONG AND MODERATE CYP3A4 INHIBITORS/DEFLAZACORT
- SLT STRONG 3A4 INHIBITORS/SILDENAFIL(PAH);TADALAFIL(BPH,PAH)
- STRONG CYP3A4 INHIBITORS/VENETOCLAX
- STRONG CYP3A4 INHIBITORS/VEMURAFENIB
- STRONG CYP3A4 INHIBITORS/TRABECTEDIN
- STRONG CYP3A4 INHIBITORS; PROTEASE INHIBITORS/CARIPRAZINE
- SELECTED P-GP INHIBITORS/EDOXABAN (> 30 MG)
- STRONG CYP3A4 INHIB;ATAZANAV;DARUNAVIR/BEDAQUILINE;DELAMANID
- SLT STRONG CYP3A4 INHIBITOR & SUBSTRATE/LUMACAFTOR-IVACAFTOR
- STRONG CYP3A4 INHIBITORS/TRASTUZUMAB EMTANSINE
- STRONG 3A4 INHIBITORS/ESZOPICLONE > 2 MG; ZOPICLONE > 5 MG
- STRONG CYP3A4 INHIBITORS/DACLATASVIR
- STRONG & MODERATE CYP3A4 INHIBITORS/ELIGLUSTAT
- STRONG UGT1A1 INHIBITORS/BELINOSTAT
- STRONG CYP3A4 INHIBITORS; PROTEASE INHIBITORS/VORAPAXAR
- STRONG & MODERATE CYP3A4 INHIBITORS/GUANFACINE
- STRONG OR MODERATE CYP3A4 INHIBITORS/SIMEPREVIR
- STRONG CYP3A4 INHIBITORS/MACITENTAN
- DUAL STRONG CYP3A4 INHIBITOR & P-GP INHIBITORS/RIOCIGUAT
- STRONG CYP3A4 INHIBITORS/QUETIAPINE
- STRONG AND MODERATE CYP3A4 INHIBITORS/BOSENTAN
- P-GP AND STRONG CYP3A4 INHIBITORS/APIXABAN
- STRONG CYP3A4 INHIBITORS/REGORAFENIB
- STRONG CYP3A4 INHIBITORS; AMPRENAVIR;ATAZANAVIR/MIFEPRISTONE
- STRONG AND MODERATE CYP3A4 INHIBITORS/IVACAFTOR
- DRONEDARONE, KETOCONAZOLE/DABIGATRAN
- SELECTED STRONG CYP3A4 INHIBITORS/SALMETEROL
- FLUCONAZOLE; KETOCONAZOLE; VORICONAZOLE/CLOPIDOGREL
- STRONG CYP3A4 INHIBITORS; DARUNAVIR/EVEROLIMUS
- P-GLYCOPROTEIN (P-GP) INHIBITORS/TOPOTECAN
- STRONG CYP3A4 INHIBITORS/MARAVIROC
- SLT AZOLE ANTIFUNGALS/SELECTED ANTICONVULSANTS; BARBITURATES
- STRONG CYP3A4 INHIBITORS/COLCHICINE
- SELECTED CYP3A4 INHIBITORS/SELECTED OPIOIDS
- ITRACONAZOLE; KETOCONAZOLE/ERYTHROMYCIN; TELITHROMYCIN
- SELECTED CYP3A4 INHIBITORS/TRAZODONE
- SLT AZOLE ANTIFUNGAL; LEVOKETOCONAZ/SELECTED VINCA ALKALOIDS
- SELECTED AZOLE ANTIFUNGAL AGENTS/SELECTED IMMUNOSUPPRESSANTS
Moderate Interactions
These medications may cause some risk when taken together. Consult your healthcare professional (e.g., doctor or pharmacist) for more in formation.
- ITRACONAZOLE; KETOCONAZOLE/AGENTS AFFECTING GASTRIC PH
- AZOLE ANTIFUNGALS/SULFONYLUREAS
- KETOCONAZOLE/SUCRALFATE
- ITRACONAZOLE; KETOCONAZOLE/SELECTED CYP3A4 INHIBITORS
- ORAL ITRACONAZOLE; KETOCONAZOLE/HYOSCYAMINE
- SELECTED AZOLE ANTIFUNGALS/BOCEPREVIR; TELAPREVIR
- STRONG CYP3A4 INHIBITORS/VAMOROLONE
- STRONG AND MODERATE CYP3A4 INHIBITORS/ETRASIMOD
- SLT STRONG CYP3A4 INHIBIT/AMLODIPINE; LEVAMLODIPINE
- STRONG CYP3A4 INHIBITORS/ZURANOLONE
- STRONG CYP3A4 INHIBITORS/QUIZARTINIB
- STR CYP3A4 INHIB;ATAZAN;DARUNAV/SLT LONG-ACTING ARIPIPRAZOLE
- STRONG CYP3A4 INHIBITORS/BORTEZOMIB
- STRONG CYP3A4 INHIBITORS/VALBENAZINE (=< 40 MG)
- STRONG CYP3A4 INHIB; PROTEASE INHIB/LUMATEPERONE (<=10.5 MG)
- STRONG CYP3A4 INHIBITORS/GILTERITINIB
- STRONG CYP3A4 INHIBITORS/TOLTERODINE (<=1 MG OR <=2 MG ER)
- LEVOKETOCONAZOLE; KETOCONAZOLE/ETHYL ALCOHOL
- STRONG CYP3A4 INHIBITORS/UPADACITINIB (<30 MG)
- STRONG CYP3A4 INHIBITORS/IBREXAFUNGERP
- STRONG CYP3A4 INHIBITORS/REPAGLINIDE
- STRONG OR MODERATE CYP2D6 OR CYP3A4 INHIBITORS/OLICERIDINE
- STRONG CYP3A4 INHIBITORS/FOSTAMATINIB
- STRONG CYP3A4 INHIBITORS/OSILODROSTAT
- SELECTED STRONG CYP3A4 INHIBITORS/ROMIDEPSIN
- STRONG CYP3A4 INHIBITORS/CANNABIDIOL-TETRAHYDROCANNABINOL
- STRONG CYP3A4 INHIBITORS/ZANUBRUTINIB
- DUAL P-GP AND STRONG CYP3A4 INHIBITORS/DAROLUTAMIDE
- SELECTED STRONG CYP3A4 INHIBITORS;PROTEASE INHIB/ILOPERIDONE
- STRONG CYP3A4 INHIBITORS; PROTEASE INHIBITORS/BREXPIPRAZOLE
- SELECTED P-GP INHIBITORS/EDOXABAN (<= 30 MG)
- STRONG CYP3A4 INHIBITORS/CLONAZEPAM
- STRONG CYP3A4 INHIBITORS/MIDOSTAURIN
- STR CYP3A4 INHIBITORS;PROTEASE INHIB/PIMAVANSERIN (<= 10 MG)
- SELECTED CYP3A4 INHIBITORS/BROMOCRIPTINE; CABERGOLINE
- P-GP AND SELECTED CYP3A4 INHIBITORS/NINTEDANIB
- STRONG 3A4 INHIB/LEVOMILNACIPRAN(<=80MG);VILAZODONE(<=20MG)
- P-GLYCOPROTEIN (P-GP) INHIBITORS/AFATINIB
- KETOCONAZOLE/FINGOLIMOD
- SELECTED CYP3A4 INHIBITORS/VARDENAFIL (<= 5 MG)
- ITRACONAZOLE;KETOCONAZOLE/SELECT BENZODIAZEPINES; BUSPIRONE
- STRONG CYP3A4 INHIBITORS/PANOBINOSTAT (<= 10 MG)
- STRONG CYP3A4 INHIB;ATAZANAV;DARUNAVIR/SAXAGLIPTIN(<=2.5 MG)
- SLT STRONG CYP3A4 INHIBIT/SELECTED CALCIUM CHANNEL BLOCKERS
- SLT AZOLE ANTIFUNGALS; LEVOKETOCONAZOLE/GEFITINIB; IMATINIB
- UGT INHIBITORS/LORAZEPAM; MEXAZOLAM
- CYP3A4; CYP2C8; P-GLYCOPROTEIN (P-GP) INHIBITORS/LOPERAMIDE
- SELECTED AZOLE ANTIFUNGAL AGENTS/SELECTED CORTICOSTEROIDS
- SELECTED AZOLE ANTIFUNGALS; LEVOKETOCONAZOLE/BUSULFAN
- STRONG CYP3A4 INHIBITORS/ESZOPICLONE; ZOPICLONE; ZOLPIDEM
- STRONG CYP3A4 INHIBITORS/CINACALCET
- KETOCONAZOLE/TIRILAZAD
- STRONG CYP3A4 INHIBITORS; ATAZANAVIR; DARUNAVIR/ARIPIPRAZOLE
- STRONG CYP3A4 INHIB; PROTEASE INHIB/ARTEMETHER;LUMEFANTRINE
- SELECTED CYP2C9 INHIBITORS/SELECTED NSAIDS
- STRONG CYP3A4 INHIBITORS/SLT LOW STRENGTH ANTIMUSCARINICS
- ITRACONAZOLE; KETOCONAZOLE/INDINAVIR
- SLT STRONG & MODERATE CYP3A4 INHIBITORS/CILOSTAZOL (<=50MG)
- SLT STRONG CYP3A4 INHIBITORS/SILDENAFIL (ED); TADALAFIL (ED)
- SELECTED P-GLYCOPROTEIN (P-GP) INHIBITORS/ETOPOSIDE
Selected from data included with permission and copyrighted by First Databank, Inc. This copyrighted material has been downloaded from a licensed data provider and is not for distribution, except as may be authorized by the applicable terms of use.
CONDITIONS OF USE: The information in this database is intended to supplement, not substitute for, the expertise and judgment of healthcare professionals. The information is not intended to cover all possible uses, directions, precautions, drug interactions or adverse effects, nor should it be construed to indicate that use of a particular drug is safe, appropriate or effective for you or anyone else. A healthcare professional should be consulted before taking any drug, changing any diet or commencing or discontinuing any course of treatment.