Does Leflunomide (Bulk) 100 % Powder Interact with other Medications?
Severe Interactions
These medications are not usually taken together. Consult your healthcare professional (e.g., doctor or pharmacist) for more in formation.
- SELECTED IMMUNOSUPPRESSANTS/NADOFARAGENE FIRADENOVEC
- WEAK CYP3A4 INHIBITORS/LEMBOREXANT (> 5 MG)
- LEFLUNOMIDE; TERIFLUNOMIDE/ROSUVASTATIN (> 10 MG)
- WEAK CYP3A4 INHIBITORS/LOMITAPIDE (>30 MG)
- SELECTED IMMUNOSUPPRESSANTS/TALIMOGENE LAHERPAREPVEC
- SELECTED IMMUNOSUPPRESSIVE AGENTS/LIVE VACCINES; LIVE BCG
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/EFALIZUMAB; NATALIZUMAB
Serious Interactions
These medications may interact and cause very harmful effects. Consult your healthcare professional (e.g., doctor or pharmacist) for more in formation.
- LEFLUNOMIDE; TERIFLUNOMIDE/BILE ACID SEQUESTRANTS
- LEFLUNOMIDE; TERIFLUNOMIDE/SELECTED IMMUNOSUPPRESSANTS
- MODERATE CYP2C8 INHIBITORS/TOVORAFENIB
- IMMUNOSUPPRESSIVE CYP2C8 INHIBITORS/PACLITAXEL
- MYELOSUPPRESSIVE MOD-WEAK 3A4 INH/SIROLIMUS PROTEIN-BOUND
- MYELOSUPPRESSIVE MOD-WEAK CYP3A4 INH/TACROLIMUS
- IMMUNOSUPPRESSIVE CYP2C8 INHIBITORS/ETRASIMOD
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/RITLECITINIB
- OATP1B3 INHIBITORS/ZAVEGEPANT
- SELECTED INHIBITORS OF BCRP WITH MYELOSUPPRESSION/CLADRIBINE
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/SIPONIMOD
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/OZANIMOD
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/FINGOLIMOD
- MYELOSUPPRESSIVES; IMMUNOMODULATORS/SODIUM IODIDE I 131
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/FILGOTINIB
- OATP1B1-3 INHIBITORS/BRINCIDOFOVIR
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/PONESIMOD
- WEAK CYP3A4 INHIBITORS/LONAFARNIB
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/BARICITINIB
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/INEBILIZUMAB
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/UPADACITINIB
- WEAK CYP3A4 INHIBITORS/ELIGLUSTAT
- SELECTED INHIBITORS OF P-GP OR BCRP/PAZOPANIB
- OATP1B1 INHIBITORS/ELUXADOLINE
- SELECTED MYELOSUPPRESSIVE AGENTS/CLOZAPINE
- WEAK CYP3A4 INHIBITORS/LOMITAPIDE (<=30MG)
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/TOFACITINIB
- SELECTED MYELOSUPPRESSIVE AGENTS/DEFERIPRONE
Moderate Interactions
These medications may cause some risk when taken together. Consult your healthcare professional (e.g., doctor or pharmacist) for more in formation.
- LEFLUNOMIDE; TERIFLUNOMIDE/METHOTREXATE (LOW STR INJ, ORAL)
- LEFLUNOMIDE/RIFAMPIN
- MODERATE CYP2C8 INHIBITORS/RESMETIROM
- MODERATE CYP2C8 INHIBITORS/DAPRODUSTAT
- OATP1B1-3 INHIBITORS/ATOGEPANT
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/COVID-19 VACCINES
- SELECTED CYP1A2 INDUCERS/OLANZAPINE-SAMIDORPHAN
- IMMUNOSUPPRESSIVES; IMMUNOMODULATORS/USTEKINUMAB
- WEAK CYP3A4 INHIBITORS/UBROGEPANT
- WEAK CYP3A4 INHIBITORS/LEMBOREXANT (<= 5 MG)
- MODERATE CYP2C8 INHIBITORS/SELEXIPAG
- SELECTED CYP1A2 INDUCERS/OLANZAPINE
- LEFLUNOMIDE; TERIFLUNOMIDE/ROSUVASTATIN (<= 10 MG)
- LEFLUNOMIDE; TERIFLUNOMIDE/SELECTED CYP2C8 SUBSTRATES
- LEFLUNOMIDE/WARFARIN
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CONDITIONS OF USE: The information in this database is intended to supplement, not substitute for, the expertise and judgment of healthcare professionals. The information is not intended to cover all possible uses, directions, precautions, drug interactions or adverse effects, nor should it be construed to indicate that use of a particular drug is safe, appropriate or effective for you or anyone else. A healthcare professional should be consulted before taking any drug, changing any diet or commencing or discontinuing any course of treatment.