Does Sustiva Interact with other Medications?
Severe Interactions
These medications are not usually taken together. Consult your healthcare professional (e.g., doctor or pharmacist) for more in formation.
- EFAVIRENZ/ST. JOHN'S WORT
- STRONG & MODERATE CYP2C19 INHIBITORS/MAVACAMTEN
- STRONG AND MODERATE CYP3A4 INDUCERS/LONAFARNIB
- EFAVIRENZ; NEVIRAPINE/ASUNAPREVIR
- STRONG & MOD 2C19 INHIB THAT PROLONG QT/CILOSTAZOL (> 50 MG)
- EFAVIRENZ; NEVIRAPINE/ELVITEGRAVIR
- STRONG CYP3A4 INDUCERS/ELBASVIR-GRAZOPREVIR
- EFAVIRENZ/PARITAPREVIR-RITONAVIR
- NNRTIS/COBICISTAT-ELVITEGRAVIR
Serious Interactions
These medications may interact and cause very harmful effects. Consult your healthcare professional (e.g., doctor or pharmacist) for more in formation.
- SELECTED PROTEASE INHIBITORS AND NNRTIS/GARLIC
- EFAVIRENZ/CARBAMAZEPINE
- EFAVIRENZ/PHENYTOIN
- EFAVIRENZ/BARBITURATES
- ANTI-RETROVIRALS/ATIDARSAGENE AUTOTEMCEL
- MODERATE CYP3A4 INDUCERS/PRAZIQUANTEL
- EFAVIRENZ/LEMBOREXANT
- P-GLYCOPROTEIN (P-GP) INDUCERS/VINCRISTINE
- ANTI-RETROVIRALS/LOVOTIBEGLOGENE AUTOTEMCEL
- STRONG AND MODERATE CYP3A4 INDUCERS/NIROGACESTAT
- STRONG OR MODERATE CYP3A4 INDUCERS/REPOTRECTINIB
- STRONG AND MODERATE CYP3A4 INDUCERS/CAPIVASERTIB
- MODERATE CYP3A4 INDUCERS/FRUQUINTINIB
- CYP3A4 INDUCERS/ZURANOLONE
- MODERATE CYP3A4 INDUCERS/PRALSETINIB
- STRONG & MODERATE CYP3A4 INDUCER THAT PROLONG QT/QUIZARTINIB
- EFAVIRENZ/VALOCTOCOGENE ROXAPARVOVEC
- STRONG & MODERATE CYP3A4 INDUCERS/SONIDEGIB
- STRONG & MODERATE CYP3A4 INDUCERS/PALBOCICLIB
- STRONG & MODERATE CYP3A4 INDUCERS/OLAPARIB
- CYP3A4 INDUCERS/ERLOTINIB
- STRONG AND MODERATE CYP3A4 INDUCERS/PALOVAROTENE
- STRONG & MODERATE CYP3A4 INDUCERS/AXITINIB
- MODERATE CYP3A4 INDUCERS/ZANUBRUTINIB
- STRONG AND MODERATE CYP3A4 INDUCERS/LENIOLISIB
- STRONG AND MODERATE CYP3A4 INDUCERS/OMAVELOXOLONE
- MODERATE CYP3A4 INDUCERS/PIRTOBRUTINIB
- STRONG AND MODERATE CYP3A4 INDUCERS/ELACESTRANT
- STRONG AND MODERATE CYP3A4 INDUCERS/CARIPRAZINE
- MODERATE CYP3A4 INDUCERS/LENACAPAVIR
- STRONG AND MODERATE CYP3A4 INDUCERS/OLUTASIDENIB
- ANTI-RETROVIRALS/ELIVALDOGENE AUTOTEMCEL
- ANTI-RETROVIRALS; HYDROXYUREA/BETIBEGLOGENE AUTOTEMCEL
- STR OR MOD 3A4 INDUC PROL QT/VONOPRAZAN-CLARITHROMYCIN-AMOX
- STRONG OR MODERATE CYP3A4 INDUCERS/VONOPRAZAN
- STRONG OR MODERATE CYP3A4 INDUCERS/GANAXOLONE
- MODERATE CYP3A4 INDUCERS THAT PROLONG QT/PACRITINIB
- POSSIBLE QT PROLONGING AGENTS/LEVOKETOCONAZOLE
- MODERATE CYP3A4 INDUCERS/DUVELISIB
- STRONG OR MODERATE CYP3A4 INDUCERS/AVACOPAN
- CYP3A4 INDUCERS/ATOGEPANT
- STRONG OR MODERATE 3A4 INDUCERS THAT PROLONG QT/MOBOCERTINIB
- STRONG & MODERATE CYP3A4 INDUCERS THAT PROLONG QT/SIPONIMOD
- STRONG & MODERATE 3A4 INDUCERS THAT PROLONG QT/FEXINIDAZOLE
- STRONG AND MODERATE CYP3A4 INDUCERS/FINERENONE
- MODERATE CYP3A4 INDUCERS/RIPRETINIB
- STRONG AND MODERATE CYP3A4 INDUCERS/IBREXAFUNGERP
- STRONG AND MODERATE CYP3A4 INDUCERS/INFIGRATINIB
- STRONG AND MOD CYP3A4 INDUCERS THAT PROLONG QT/PIMAVANSERIN
- STRONG & MOD CYP3A4 INDUCERS THAT PROLONG QT/BEDAQUILINE
- STRONG AND MOD CYP3A4 INDUCERS THAT PROLONG QT/SELPERCATINIB
- STRONG OR MODERATE CYP3A4 INDUCERS THAT PROLONG QT/LEFAMULIN
- STRONG AND MOD CYP3A4 INDUCERS THAT PROLONG QT/ENTRECTINIB
- STRONG AND MOD CYP3A4 INDUCERS THAT PROLONG QT/GLASDEGIB
- MODERATE CYP3A4 INDUCERS THAT PROLONG QT/CRIZOTINIB
- STRONG AND MODERATE CYP3A4 INDUCERS/VOCLOSPORIN
- MODERATE CYP3A4 INDUCERS/IDELALISIB
- SELECTED P-GP INDUCERS/BEROTRALSTAT
- STRONG AND MODERATE CYP3A4 INDUCERS/CAPMATINIB
- UGT1A1 INDUCERS/SACITUZUMAB GOVITECAN
- STRONG AND MODERATE CYP3A4 INDUCERS/PEMIGATINIB
- STRONG AND MODERATE CYP3A4 INDUCERS/SELUMETINIB
- STRONG AND MODERATE CYP3A4 INDUCERS/RIMEGEPANT
- STRONG OR MODERATE CYP3A4 INDUCERS/TAZEMETOSTAT
- MODERATE CYP3A4 INDUCERS/IBRUTINIB
- STRONG OR MODERATE CYP3A4 INDUCERS/AVAPRITINIB
- CYP3A4 INDUCERS/LUMATEPERONE
- STRONG OR MODERATE CYP3A4 INDUCERS/DARIDOREXANT
- SELECTED STRONG OR MODERATE CYP3A4 INDUCERS/VOXELOTOR
- P-GLYCOPROTEIN (P-GP) OR UGT INDUCERS/LETERMOVIR
- MODERATE CYP3A4 INDUCERS/FEDRATINIB
- STRONG AND MODERATE CYP3A4 INDUCERS/PRETOMANID
- P-GP AND MODERATE CYP3A4 INDUCERS/DAROLUTAMIDE
- MODERATE CYP3A4 INDUCERS/ERDAFITINIB
- MODERATE CYP3A4 INDUCERS/BRIGATINIB
- MODERATE CYP3A4 INDUCERS/LORLATINIB
- EFAVIRENZ;ETRAVIRINE;NEVIRAPINE/DORAVIRINE
- MODERATE CYP3A4 INDUCERS/ABEMACICLIB
- STRONG 2C19 AND 3A4 INDUCERS/SLT PROTON PUMP INHIBITORS
- STRONG AND MODERATE CYP3A4 INDUCERS/NERATINIB
- P-GLYCOPROTEIN (P-GP) INDUCERS/ETOPOSIDE
- MODERATE CYP3A4 INDUCERS/VENETOCLAX
- SELECTED ANTIRETROVIRALS/ORLISTAT
- EFAVIRENZ/ATOVAQUONE; PROGUANIL
- EFAVIRENZ;ETRAVIRINE;NEVIRAPINE/COBICISTAT-BOOSTED DARUNAVIR
- EFAVIRENZ/ARTEMETHER; LUMEFANTRINE
- SELECT CYP2C19 AND CYP3A4 INDUCER/ESOMEPRAZOLE; OMEPRAZOLE
- STRONG & MODERATE CYP3A4 INDUCERS/GUANFACINE
- ETRAVIRINE; EFAVIRENZ; NEVIRAPINE/DOLUTEGRAVIR
- UGT INDUCERS/CANAGLIFLOZIN
- EFAVIRENZ; ETRAVIRINE;NEVIRAPINE/SELECTED HEPATITIS C AGENTS
- STRONG & MODERATE CYP3A4 INDUCERS/COBIMETINIB
- P-GP & STRONG 3A4 INDUCERS;EFAVIRENZ;PB/APIXABAN;RIVAROXABAN
- STRONG P-GP OR CYP3A4 INDUCER/LINAGLIPTIN
- EFAVIRENZ; ETRAVIRINE/CLOPIDOGREL
- STRONG UGT INDUCERS/DEFERASIROX
- EFAVIRENZ/ATAZANAVIR
- STRONG CYP3A4 INDUCERS/MARAVIROC
- EFAVIRENZ/ITRACONAZOLE; KETOCONAZOLE; POSACONAZOLE
- SELECTED QT PROLONGING AGENTS/ZIPRASIDONE
- EFAVIRENZ/VORICONAZOLE
- EFAVIRENZ/FOSAMPRENAVIR; SAQUINAVIR
- EFAVIRENZ/INDINAVIR
- EFAVIRENZ; NEVIRAPINE/HORMONAL CONTRACEPTIVE AGENTS
Moderate Interactions
These medications may cause some risk when taken together. Consult your healthcare professional (e.g., doctor or pharmacist) for more in formation.
- EFAVIRENZ/QT PROLONGING AGENTS
- SENSITIVE CYP2B6 SUBSTRATES THAT PROLONG QT/MIDOSTAURIN
- POSSIBLE QT PROLONGING AGENTS/DEXMEDETOMIDINE SUBLINGUAL
- QT PROLONGING AGENTS/ETRASIMOD
- QT PROLONGING AGENTS/GEPIRONE
- STRONG AND MODERATE CYP3A4 INDUCERS/SILDENAFIL (PAH)
- POSSIBLE QT PROLONGING AGENTS/ADAGRASIB
- MODERATE CYP3A4 INDUCERS/LAROTRECTINIB
- QT PROLONGING AGENTS/TUCIDINOSTAT
- MODERATE CYP2B6 INDUCERS/BUPROPION COMBINATIONS
- MODERATE AND WEAK CYP3A4 INDUCERS THAT PROLONG QT/TACROLIMUS
- QT PROLONGING AGENTS/SAVOLITINIB
- QT PROLONGING AGENTS/TRICLABENDAZOLE
- POSSIBLE QT PROLONGING AGENTS/PANOBINOSTAT
- QT PROLONGING AGENTS/OZANIMOD
- QT PROLONGING AGENTS/PONESIMOD
- QT PROLONGING AGENTS/GALANTAMINE
- SLT 2C19&3A4 INDUCER THAT PROLONG QT/CITALOPRAM;ESCITALOPRAM
- STRONG UGT INDUCERS; NEVIRAPINE/ARTESUNATE
- QT PROLONGING AGENTS/OSILODROSTAT
- QT PROLONGING AGENTS/AMISULPRIDE
- MODERATE CYP3A4 INDUCERS/ROLAPITANT
- MODERATE AND WEAK CYP3A4 INDUCERS/UBROGEPANT
- POSSIBLE QT PROLONGING AGENTS/HYDROXYCHLOROQUINE
- SELECTED UGT AND STRONG CYP3A4 INDUCERS/OXCARBAZEPINE
- POSSIBLE QT PROLONGING AGENTS/ENCORAFENIB
- STRONG AND MODERATE CYP3A4 INDUCERS/PERAMPANEL
- POSSIBLE QT PROLONGING AGENTS/RIBOCICLIB
- MODERATE CYP3A4 INDUCERS/DACLATASVIR
- SELECTED MODERATE-WEAK CYP3A4 INDUCERS/EXEMESTANE
- P-GLYCOPROTEIN (P-GP) INDUCERS; PHENOBARBITAL/AFATINIB
- QT PROLONGING AGENTS/FINGOLIMOD
- MODERATE CYP2B6 INDUCERS/BUPROPION
- POSSIBLE QT PROLONGING AGENTS/GADOFOSVESET
- NNRTIS/CLARITHROMYCIN
- EFAVIRENZ; NEVIRAPINE/LEVOMETHADONE; METHADONE
- EFAVIRENZ/RIFABUTIN
- EFAVIRENZ; NEVIRAPINE/CASPOFUNGIN
- EFAVIRENZ; NEVIRAPINE/LOPINAVIR
- STRONG & MOD 2C19 INHIB THAT PROLONG QT/CILOSTAZOL (<=50MG)
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CONDITIONS OF USE: The information in this database is intended to supplement, not substitute for, the expertise and judgment of healthcare professionals. The information is not intended to cover all possible uses, directions, precautions, drug interactions or adverse effects, nor should it be construed to indicate that use of a particular drug is safe, appropriate or effective for you or anyone else. A healthcare professional should be consulted before taking any drug, changing any diet or commencing or discontinuing any course of treatment.